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Bioorganic and medicinal Chemistry
Bioorganic and medicinal Chemistry
Novel pyrazolopyrimidine derivatives as GSK-3 inhibitors
Organic Chemistry / Enzyme Inhibitors / Tight Binding / Bioorganic and medicinal Chemistry / Pyrazoles
Peptide-based hydrogel nanoparticles as effective drug delivery agents
Organic Chemistry / Nanoparticles / Hydrogel / Peptides / Drug Delivery Systems / Particle Size / Surface Properties / Bioorganic and medicinal Chemistry / Drug Carriers / Particle Size / Surface Properties / Bioorganic and medicinal Chemistry / Drug Carriers
Synthetic mannosides act as acceptors for mycobacterial α1-6 mannosyltransferase
Organic Chemistry / Mass Spectrometry / Gas Chromatography/mass Spectrometry / Bioorganic and medicinal Chemistry / Thin Layer Chromatography / Bioorganic / Linkage Analysis / Bioorganic / Linkage Analysis
Hydrolase and sialyltransferase activities of Trypanosoma cruzi trans-sialidase towards NeuAc-α-2,3-Gal-β-O-PNP
Organic Chemistry / Glycoproteins / Neuraminidase / Trypanosoma Cruzi / Substrate Specificity / Spectrum analysis / Bioorganic and medicinal Chemistry / Disaccharides / Clostridium perfringens / Trans-Sialidase / Glycosyl Hydrolases / Spectrum analysis / Bioorganic and medicinal Chemistry / Disaccharides / Clostridium perfringens / Trans-Sialidase / Glycosyl Hydrolases
Synthetic mannosides act as acceptors for mycobacterial a1-6 mannosyltransferase
Organic Chemistry / Mass Spectrometry / Gas Chromatography/mass Spectrometry / Bioorganic and medicinal Chemistry / Thin Layer Chromatography / Linkage Analysis
7-Methoxyfuro[2,3-c]pyridine-4-carboxamides as PDE4 Inhibitors: A Potential Treatment for Asthma
Organic Chemistry / Animals / Phosphodiesterase Inhibitors / Pyridines / Bioorganic and medicinal Chemistry / Structure activity Relationship / Furans / Structure activity Relationship / Furans
Polyacylated neohesperidosides From Geranium caespitosum: bacterial multidrug resistance pump inhibitors
Organic Chemistry / Pharmacognosy / Structural Analysis / Multidrug Resistance / Resistance / Bacteria / Staphylococcus aureus / Membrane transport proteins / Isolation / Anti-Bacterial Agents / Bacillus subtilis / Bacillus megaterium / Microbial Sensitivity Tests / Acylation / Bioorganic and medicinal Chemistry / Biological activity / Drug Interaction / Hesperidin / Geranium / Bacteria / Staphylococcus aureus / Membrane transport proteins / Isolation / Anti-Bacterial Agents / Bacillus subtilis / Bacillus megaterium / Microbial Sensitivity Tests / Acylation / Bioorganic and medicinal Chemistry / Biological activity / Drug Interaction / Hesperidin / Geranium
Biphenyl derivatives as novel dual NK1/NK2-receptor antagonists
Organic Chemistry / Humans / Animals / Conformational Analysis / Molecular Conformation / Bioorganic and medicinal Chemistry / Biological activity / Structure activity Relationship / Molecular Structure / Neurokinin receptor antagonists / Bioorganic and medicinal Chemistry / Biological activity / Structure activity Relationship / Molecular Structure / Neurokinin receptor antagonists
Novel IKK inhibitors: beta-carbolines
Organic Chemistry / Enzyme Inhibitors / Western blotting / Humans / HeLa cells / Bioorganic and medicinal Chemistry / Structure activity Relationship / Bioorganic and medicinal Chemistry / Structure activity Relationship
Novel IKK inhibitors: beta-carbolines
Organic Chemistry / Enzyme Inhibitors / Western blotting / Humans / HeLa cells / Bioorganic and medicinal Chemistry / Structure activity Relationship / Bioorganic and medicinal Chemistry / Structure activity Relationship
Novel IKK inhibitors: beta-carbolines
Organic Chemistry / Enzyme Inhibitors / Western blotting / Humans / HeLa cells / Bioorganic and medicinal Chemistry / Structure activity Relationship / Bioorganic and medicinal Chemistry / Structure activity Relationship
Novel IKK inhibitors: beta-carbolines
Organic Chemistry / Enzyme Inhibitors / Western blotting / Humans / HeLa cells / Bioorganic and medicinal Chemistry / Structure activity Relationship / Bioorganic and medicinal Chemistry / Structure activity Relationship
Oximinoarylsulfonamides as potent HIV protease inhibitors
Organic Chemistry / Kinetics / HIV protease / Drug Design / Molecular Conformation / Bioorganic and medicinal Chemistry / Structure activity Relationship / Carbamates / Bioorganic and medicinal Chemistry / Structure activity Relationship / Carbamates
Discovery of ectoparasiticidal hydrazonotrifluoromethanesulfonanilides
Organic Chemistry / Drug Discovery / Cats / Dogs / Animals / Hydrazones / Bioorganic and medicinal Chemistry / Structure activity Relationship / Rhipicephalus sanguineus / Hydrazones / Bioorganic and medicinal Chemistry / Structure activity Relationship / Rhipicephalus sanguineus
Novel IKK inhibitors: beta-carbolines
Organic Chemistry / Enzyme Inhibitors / Western blotting / Humans / HeLa cells / Bioorganic and medicinal Chemistry / Structure activity Relationship / Bioorganic and medicinal Chemistry / Structure activity Relationship
Inhibition of phospho-MurNAc-pentapeptide translocase (MraY) by nucleoside natural product antibiotics, bacteriophage ϕX174 lysis protein E, and cationic antibacterial peptides
Organic Chemistry / Bioorganic and medicinal Chemistry
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