Bioorganic and medicinal Chemistry

Novel pyrazolopyrimidine derivatives as GSK-3 inhibitors

Organic Chemistry / Enzyme Inhibitors / Tight Binding / Bioorganic and medicinal Chemistry / Pyrazoles

Peptide-based hydrogel nanoparticles as effective drug delivery agents

Organic Chemistry / Nanoparticles / Hydrogel / Peptides / Drug Delivery Systems / Particle Size / Surface Properties / Bioorganic and medicinal Chemistry / Drug Carriers / Particle Size / Surface Properties / Bioorganic and medicinal Chemistry / Drug Carriers

Synthetic mannosides act as acceptors for mycobacterial α1-6 mannosyltransferase

Organic Chemistry / Mass Spectrometry / Gas Chromatography/mass Spectrometry / Bioorganic and medicinal Chemistry / Thin Layer Chromatography / Bioorganic / Linkage Analysis / Bioorganic / Linkage Analysis

Hydrolase and sialyltransferase activities of Trypanosoma cruzi trans-sialidase towards NeuAc-α-2,3-Gal-β-O-PNP

Organic Chemistry / Glycoproteins / Neuraminidase / Trypanosoma Cruzi / Substrate Specificity / Spectrum analysis / Bioorganic and medicinal Chemistry / Disaccharides / Clostridium perfringens / Trans-Sialidase / Glycosyl Hydrolases / Spectrum analysis / Bioorganic and medicinal Chemistry / Disaccharides / Clostridium perfringens / Trans-Sialidase / Glycosyl Hydrolases

Synthetic mannosides act as acceptors for mycobacterial a1-6 mannosyltransferase

Organic Chemistry / Mass Spectrometry / Gas Chromatography/mass Spectrometry / Bioorganic and medicinal Chemistry / Thin Layer Chromatography / Linkage Analysis

7-Methoxyfuro[2,3-c]pyridine-4-carboxamides as PDE4 Inhibitors: A Potential Treatment for Asthma

Organic Chemistry / Animals / Phosphodiesterase Inhibitors / Pyridines / Bioorganic and medicinal Chemistry / Structure activity Relationship / Furans / Structure activity Relationship / Furans

Polyacylated neohesperidosides From Geranium caespitosum: bacterial multidrug resistance pump inhibitors

Organic Chemistry / Pharmacognosy / Structural Analysis / Multidrug Resistance / Resistance / Bacteria / Staphylococcus aureus / Membrane transport proteins / Isolation / Anti-Bacterial Agents / Bacillus subtilis / Bacillus megaterium / Microbial Sensitivity Tests / Acylation / Bioorganic and medicinal Chemistry / Biological activity / Drug Interaction / Hesperidin / Geranium / Bacteria / Staphylococcus aureus / Membrane transport proteins / Isolation / Anti-Bacterial Agents / Bacillus subtilis / Bacillus megaterium / Microbial Sensitivity Tests / Acylation / Bioorganic and medicinal Chemistry / Biological activity / Drug Interaction / Hesperidin / Geranium

Biphenyl derivatives as novel dual NK1/NK2-receptor antagonists

Organic Chemistry / Humans / Animals / Conformational Analysis / Molecular Conformation / Bioorganic and medicinal Chemistry / Biological activity / Structure activity Relationship / Molecular Structure / Neurokinin receptor antagonists / Bioorganic and medicinal Chemistry / Biological activity / Structure activity Relationship / Molecular Structure / Neurokinin receptor antagonists

Novel IKK inhibitors: beta-carbolines

Organic Chemistry / Enzyme Inhibitors / Western blotting / Humans / HeLa cells / Bioorganic and medicinal Chemistry / Structure activity Relationship / Bioorganic and medicinal Chemistry / Structure activity Relationship

Novel IKK inhibitors: beta-carbolines

Organic Chemistry / Enzyme Inhibitors / Western blotting / Humans / HeLa cells / Bioorganic and medicinal Chemistry / Structure activity Relationship / Bioorganic and medicinal Chemistry / Structure activity Relationship

Novel IKK inhibitors: beta-carbolines

Organic Chemistry / Enzyme Inhibitors / Western blotting / Humans / HeLa cells / Bioorganic and medicinal Chemistry / Structure activity Relationship / Bioorganic and medicinal Chemistry / Structure activity Relationship

Novel IKK inhibitors: beta-carbolines

Organic Chemistry / Enzyme Inhibitors / Western blotting / Humans / HeLa cells / Bioorganic and medicinal Chemistry / Structure activity Relationship / Bioorganic and medicinal Chemistry / Structure activity Relationship

Oximinoarylsulfonamides as potent HIV protease inhibitors

Organic Chemistry / Kinetics / HIV protease / Drug Design / Molecular Conformation / Bioorganic and medicinal Chemistry / Structure activity Relationship / Carbamates / Bioorganic and medicinal Chemistry / Structure activity Relationship / Carbamates

Discovery of ectoparasiticidal hydrazonotrifluoromethanesulfonanilides

Organic Chemistry / Drug Discovery / Cats / Dogs / Animals / Hydrazones / Bioorganic and medicinal Chemistry / Structure activity Relationship / Rhipicephalus sanguineus / Hydrazones / Bioorganic and medicinal Chemistry / Structure activity Relationship / Rhipicephalus sanguineus

Novel IKK inhibitors: beta-carbolines

Organic Chemistry / Enzyme Inhibitors / Western blotting / Humans / HeLa cells / Bioorganic and medicinal Chemistry / Structure activity Relationship / Bioorganic and medicinal Chemistry / Structure activity Relationship
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