Enzyme Inhibitors

Glucocorticoid receptor deficiency increases vulnerability of the nigrostriatal dopaminergic system: critical role of glial nitric oxide

Physiology / Enzyme Inhibitors / Oxidative Stress / Macrophages / Dopamine / Mice / Nitric oxide / Animals / Corticosterone / Substantia nigra / Medical Physiology / Neurons / Lysine / Nitric Oxide Synthase / Biochemistry and cell biology / Mice / Nitric oxide / Animals / Corticosterone / Substantia nigra / Medical Physiology / Neurons / Lysine / Nitric Oxide Synthase / Biochemistry and cell biology

Establishment of a cell-free system of neuronal apoptosis: comparison of premitochondrial, mitochondrial, and postmitochondrial phases

Enzyme Inhibitors / Mitochondria / Apoptosis / Neuronal cell death / Caspases / Cerebellum / Animals / Cytochrome C / Peptides / The / Neurons / Caspase / Tamoxifen / Rats / Cysteine endopeptidases / Nervous System / Cell free System / Staurosporine / Adenosine Triphosphate / DNA fragmentation / Neuronal apoptosis / Molecular Sequence Data / Cerebellum / Animals / Cytochrome C / Peptides / The / Neurons / Caspase / Tamoxifen / Rats / Cysteine endopeptidases / Nervous System / Cell free System / Staurosporine / Adenosine Triphosphate / DNA fragmentation / Neuronal apoptosis / Molecular Sequence Data

Phenoxyacetohydrazide Schiff Bases: β-Glucuronidase Inhibitors

Organic Chemistry / Enzyme Inhibitors / Animals / Glucuronidase / Schiff bases / Cattle / Molecules / Cattle / Molecules

Pyrano chalcones and a flavone from Neoraputia magnifica and their Trypanosoma cruzi glycosomal glyceraldehyde-3-phosphate dehydrogenase-inhibitory activities

Phytochemistry / Enzyme Inhibitors / Flavonoids / Biological Sciences / Animals / CHEMICAL SCIENCES / Trypanosoma Cruzi / Trypanocidal Agents / Recombinant Proteins / CHEMICAL SCIENCES / Trypanosoma Cruzi / Trypanocidal Agents / Recombinant Proteins

Design of bioavailable derivatives of 12-(3-adamantan-1-yl-ureido)dodecanoic acid, a potent inhibitor of the soluble epoxide hydrolase

Organic Chemistry / Enzyme Inhibitors / Humans / Mice / Blood Pressure / Animals / Male / Drug Design / Solubility / Time Factors / Functional Group / Bioorganic and medicinal Chemistry / Structure activity Relationship / Adamantane / Physical Properties / Molecular Structure / Animals / Male / Drug Design / Solubility / Time Factors / Functional Group / Bioorganic and medicinal Chemistry / Structure activity Relationship / Adamantane / Physical Properties / Molecular Structure

Novel indoleamine 2,3-dioxygenase-1 inhibitors from a multistep in silico screen

Organic Chemistry / Enzyme Inhibitors / Humans / Drug Design / Thiourea / Enzyme / Bioorganic and medicinal Chemistry / In Silico / Protein Binding / Enzyme / Bioorganic and medicinal Chemistry / In Silico / Protein Binding

A Novel Potent Nicotinamide Phosphoribosyltransferase Inhibitor Synthesized via Click Chemistry

Organic Chemistry / Medicinal Chemistry / Enzyme Inhibitors / Autophagy / Humans / Animals / Medicinal / Structure activity Relationship / Protein Binding / Antineoplastic Agents / Alkynes / Animals / Medicinal / Structure activity Relationship / Protein Binding / Antineoplastic Agents / Alkynes

A subgroup of pancreatic adenocarcinoma is sensitive to the 5-aza-dC DNA methyltransferase inhibitor

Enzyme Inhibitors / Transcriptome / Humans / Mice / Animals

Nebivolol Increases Arterial Distensibility In Vivo

Enzyme Inhibitors / Cardiovascular Risk / Hypertension / Hemodynamics / Sheep / Blood Pressure / Nitric oxide / Animals / Arterial stiffness / Clinical Sciences / Nitric Oxide Synthase / Pulse Wave Velocity / Nitroglycerin / Vascular Resistance / Atenolol / Blood Pressure / Nitric oxide / Animals / Arterial stiffness / Clinical Sciences / Nitric Oxide Synthase / Pulse Wave Velocity / Nitroglycerin / Vascular Resistance / Atenolol

Fragment-based design of 3-aminopyridine-derived amides as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT)

Organic Chemistry / Cytokines / Enzyme Inhibitors / Macromolecular X-Ray Crystallography / Humans / Amides / Cell Proliferation / Structure activity Relationship / Antineoplastic Agents / Amides / Cell Proliferation / Structure activity Relationship / Antineoplastic Agents

Arylfurans as potential Trypanosoma cruzi trypanothione reductase inhibitors

Medical Microbiology / Enzyme Inhibitors / Mice / Animals / Male / Chagas disease / Total Synthesis / Trypanosoma Cruzi / Trypanocidal Agents / Structure activity Relationship / Furans / Chagas disease / Total Synthesis / Trypanosoma Cruzi / Trypanocidal Agents / Structure activity Relationship / Furans

P2Y6 Nucleotide Receptor Activates PKC to Protect 1321N1 Astrocytoma Cells Against Tumor Necrosis Factor-Induced Apoptosis

Drug interactions / Enzyme Inhibitors / Apoptosis / Molecular and cellular biology / Humans / Cellular and Molecular Neurobiology / Animals / Calcium Signaling / Astrocytes / Rats / Tumor necrosis factor-alpha / Protein isoforms / Astrocytoma / Tumor Necrosis Factor–α (TNF) / Intracellular Signaling / Neurosciences / Nucleotides / Biochemistry and cell biology / Cellular and Molecular Neurobiology / Animals / Calcium Signaling / Astrocytes / Rats / Tumor necrosis factor-alpha / Protein isoforms / Astrocytoma / Tumor Necrosis Factor–α (TNF) / Intracellular Signaling / Neurosciences / Nucleotides / Biochemistry and cell biology

Tropolysin, a New Oligopeptidase from African Trypanosomes † , ‡

Biochemistry / Africa / Enzyme Inhibitors / Phylogeny / Humans / Sequence alignment / Animals / Peptides / Cattle / Trypanosoma brucei brucei / Protozoan Proteins / Amino Acid Sequence / Biochemistry and cell biology / Sequence alignment / Animals / Peptides / Cattle / Trypanosoma brucei brucei / Protozoan Proteins / Amino Acid Sequence / Biochemistry and cell biology

DIABLO Promotes Apoptosis by Removing MIHA/XIAP from Processed Caspase 9

Flow Cytometry / Enzyme Inhibitors / Cell Biology / Apoptosis / Western blotting / Biological Sciences / Saccharomyces cerevisiae / Caspases / Cell line / Humans / Uv Radiation / Cell Death / Cytochrome C / Proteins / Caspase / The cell / Transfection / Apoptotic Protease Activating Factor-1 / Mitochondrial Proteins / Biological Sciences / Saccharomyces cerevisiae / Caspases / Cell line / Humans / Uv Radiation / Cell Death / Cytochrome C / Proteins / Caspase / The cell / Transfection / Apoptotic Protease Activating Factor-1 / Mitochondrial Proteins

8-BuS-ATP derivatives as specific NTPDase1 inhibitors

Enzyme Inhibitors / Cercopithecus aethiops / Humans / Platelet aggregation / Mice / Animals / Rats / Species Specificity / Adenosine Triphosphate / Adenosine monophosphate / Adenosine Diphosphate / Animals / Rats / Species Specificity / Adenosine Triphosphate / Adenosine monophosphate / Adenosine Diphosphate

Analogs of natural aminoacyl-tRNA synthetase inhibitors clear malaria in vivo

Enzyme Inhibitors / Multidisciplinary / Humans / Mice / Animals / Plasmodium falciparum / Antimalarials / Plasmodium falciparum / Antimalarials

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