Prodrugs

Thermolytic CpG-containing DNA oligonucleotides as potential immunotherapeutic prodrugs

Cytokines / Biological Sciences / Environmental Sciences / Prodrugs / Infectious Disease / Mice / Female / Animals / Nucleic Acids / Cutaneous Leishmaniasis / Virus infection / Leishmania Major / *Hot Temperature / Mice / Female / Animals / Nucleic Acids / Cutaneous Leishmaniasis / Virus infection / Leishmania Major / *Hot Temperature

Efficacy of DA7218, a New Oxazolidinone Prodrug, in the Treatment of Experimental Actinomycetoma Produced by Nocardia brasiliensis

Organic Chemistry / Treatment Outcome / Prodrugs / Mice / Animals / Molecules / Mycetoma / Actinomycosis / Organophosphates / Nocardia / Oxazolidinones / Acetamides / Tetrazoles / Molecules / Mycetoma / Actinomycosis / Organophosphates / Nocardia / Oxazolidinones / Acetamides / Tetrazoles

Efficacy of DA7218, a New Oxazolidinone Prodrug, in the Treatment of Experimental Actinomycetoma Produced by Nocardia brasiliensis

Organic Chemistry / Treatment Outcome / Prodrugs / Mice / Animals / Molecules / Mycetoma / Actinomycosis / Organophosphates / Nocardia / Oxazolidinones / Acetamides / Tetrazoles / Molecules / Mycetoma / Actinomycosis / Organophosphates / Nocardia / Oxazolidinones / Acetamides / Tetrazoles

In Vitro Activities of DA7157 and DA7218 against Mycobacterium tuberculosis and Nocardia brasiliensis

Microbiology / Medical Microbiology / Tuberculosis / Prodrugs / Humans / Mycobacterium tuberculosis / Multidrug Resistance / Anti-Bacterial Agents / Antimicrobial agents / Microbial Sensitivity Tests / Mycetoma / Organophosphates / Nocardia / Oxazolidinones / Tetrazoles / Mycobacterium tuberculosis / Multidrug Resistance / Anti-Bacterial Agents / Antimicrobial agents / Microbial Sensitivity Tests / Mycetoma / Organophosphates / Nocardia / Oxazolidinones / Tetrazoles

Efficacy of DA-7218, a New Oxazolidinone Prodrug, in the Treatment of Experimental Actinomycetoma Produced by Nocardia brasiliensis

Organic Chemistry / Treatment Outcome / Prodrugs / Mice / Animals / Molecules / Mycetoma / Actinomycosis / Organophosphates / Nocardia / Oxazolidinones / Acetamides / Tetrazoles / Molecules / Mycetoma / Actinomycosis / Organophosphates / Nocardia / Oxazolidinones / Acetamides / Tetrazoles

Dimeric l-Dopa Derivatives as Potential Prodrugs

Organic Chemistry / Kinetics / In Vitro / Prodrugs / Humans / Animals / Plasma / Prodrug / Partition Coefficient / Levodopa / Shell Half-Life / Rats / Rat / Aqueous Solution / Hydrolysis / Chemical Stability / Drug Stability / Hydrogen-Ion Concentration / Chemical Synthesis / Physicochemical Properties / Dimerization / Enantiomer / Animals / Plasma / Prodrug / Partition Coefficient / Levodopa / Shell Half-Life / Rats / Rat / Aqueous Solution / Hydrolysis / Chemical Stability / Drug Stability / Hydrogen-Ion Concentration / Chemical Synthesis / Physicochemical Properties / Dimerization / Enantiomer

Dimeric l-Dopa Derivatives as Potential Prodrugs

Organic Chemistry / Kinetics / In Vitro / Prodrugs / Humans / Animals / Plasma / Prodrug / Partition Coefficient / Levodopa / Shell Half-Life / Rats / Rat / Aqueous Solution / Hydrolysis / Chemical Stability / Drug Stability / Hydrogen-Ion Concentration / Chemical Synthesis / Physicochemical Properties / Dimerization / Enantiomer / Animals / Plasma / Prodrug / Partition Coefficient / Levodopa / Shell Half-Life / Rats / Rat / Aqueous Solution / Hydrolysis / Chemical Stability / Drug Stability / Hydrogen-Ion Concentration / Chemical Synthesis / Physicochemical Properties / Dimerization / Enantiomer

Synthesis of l-(+)-3-(3-hydroxy-4-pivaloyloxybenzyl)-2,5-diketomorpholine as potential prodrug of l-dopa

Organic Chemistry / Prodrugs / Humans / Animals / Levodopa / Shell Half-Life / Rats / Shell Half-Life / Rats

Dimeric l-Dopa Derivatives as Potential Prodrugs

Organic Chemistry / Kinetics / In Vitro / Prodrugs / Humans / Animals / Plasma / Prodrug / Partition Coefficient / Levodopa / Shell Half-Life / Rats / Rat / Aqueous Solution / Hydrolysis / Chemical Stability / Drug Stability / Hydrogen-Ion Concentration / Chemical Synthesis / Physicochemical Properties / Dimerization / Enantiomer / Animals / Plasma / Prodrug / Partition Coefficient / Levodopa / Shell Half-Life / Rats / Rat / Aqueous Solution / Hydrolysis / Chemical Stability / Drug Stability / Hydrogen-Ion Concentration / Chemical Synthesis / Physicochemical Properties / Dimerization / Enantiomer

Thermolytic CpG-containing DNA oligonucleotides as potential immunotherapeutic prodrugs

Cytokines / Biological Sciences / Environmental Sciences / Prodrugs / Infectious Disease / Mice / Female / Animals / Nucleic Acids / Cutaneous Leishmaniasis / Virus infection / Leishmania Major / *Hot Temperature / Mice / Female / Animals / Nucleic Acids / Cutaneous Leishmaniasis / Virus infection / Leishmania Major / *Hot Temperature

Thermolytic CpG-containing DNA oligonucleotides as potential immunotherapeutic prodrugs

Cytokines / Biological Sciences / Environmental Sciences / Prodrugs / Infectious Disease / Mice / Female / Animals / Nucleic Acids / Cutaneous Leishmaniasis / Virus infection / Leishmania Major / *Hot Temperature / Mice / Female / Animals / Nucleic Acids / Cutaneous Leishmaniasis / Virus infection / Leishmania Major / *Hot Temperature

In Vitro Activities of DA-7157 and DA-7218 against Mycobacterium tuberculosis and Nocardia brasiliensis

Microbiology / Medical Microbiology / Tuberculosis / Prodrugs / Humans / Mycobacterium tuberculosis / Multidrug Resistance / Anti-Bacterial Agents / Antimicrobial agents / Microbial Sensitivity Tests / Mycetoma / Organophosphates / Nocardia / Oxazolidinones / Mycobacterium tuberculosis / Multidrug Resistance / Anti-Bacterial Agents / Antimicrobial agents / Microbial Sensitivity Tests / Mycetoma / Organophosphates / Nocardia / Oxazolidinones

Efficacy of DA-7218, a New Oxazolidinone Prodrug, in the Treatment of Experimental Actinomycetoma Produced by Nocardia brasiliensis

Organic Chemistry / Treatment Outcome / Prodrugs / Mice / Animals / Molecules / Mycetoma / Actinomycosis / Organophosphates / Nocardia / Oxazolidinones / Acetamides / Molecules / Mycetoma / Actinomycosis / Organophosphates / Nocardia / Oxazolidinones / Acetamides

IMP - GMP specific cytosolic 5\'-nucleotidase regulates nucleotide pool and prodrug metabolism

Biological Sciences / Prodrugs / Humans / Drug Resistance / Physical sciences / Phosphorylation / Substrate Specificity / Cell Survival / Antineoplastic Agents / Nucleotides / Immunoblotting / Phosphorylation / Substrate Specificity / Cell Survival / Antineoplastic Agents / Nucleotides / Immunoblotting

Human Neural Stem Cell Tropism to Metastatic Breast Cancer

Technology / Stem Cells / Biological Sciences / Prodrugs / Humans / Mice / Female / Animals / STEM / Drug Delivery Systems / Neoplasm Invasiveness / Biotransformation / Neural Stem Cells / Camptothecin / Rabbits / Cell Survival / Interleukin / Mice / Female / Animals / STEM / Drug Delivery Systems / Neoplasm Invasiveness / Biotransformation / Neural Stem Cells / Camptothecin / Rabbits / Cell Survival / Interleukin

Synthesis of l-(+)-3-(3-hydroxy-4-pivaloyloxybenzyl)-2,5-diketomorpholine as potential prodrug of l-dopa

Organic Chemistry / Prodrugs / Humans / Animals / Levodopa / Shell Half-Life / Rats / Shell Half-Life / Rats
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