Quinolines

In Silico Studies of Quinoxaline-2-Carboxamide 1,4-di-N-Oxide Derivatives as Antimycobacterial Agents

Organic Chemistry / Cercopithecus aethiops / Mycobacterium tuberculosis / Computer Simulation / Animals / Molecules / Anti-Bacterial Agents / Quinolines / Vero cells / Molecular Structure / Molecules / Anti-Bacterial Agents / Quinolines / Vero cells / Molecular Structure

Cryptolepine, isolated from Sida acuta, sensitizes human gastric adenocarcinoma cells to TRAIL-induced apoptosis

Cancer / Apoptosis / Biological Sciences / Phytotherapy / Humans / Caspase / CHEMICAL SCIENCES / Malvaceae / Rail Trails / Quinolines / Sida Acuta / Cryptolepine / TRAIL induced Apoptosis / AGS Cell Lines / Indole Alkaloids / Glycosides / Adenocarcinoma / Caspase / CHEMICAL SCIENCES / Malvaceae / Rail Trails / Quinolines / Sida Acuta / Cryptolepine / TRAIL induced Apoptosis / AGS Cell Lines / Indole Alkaloids / Glycosides / Adenocarcinoma

Montelukast exerts no acute direct effect on NO synthases

Gene expression / Humans / Female / Animals / Male / Penis / Lung / Vasoconstriction / Clinical Sciences / Lipopolysaccharides / Rats / Wistar Rats / Rabbits / Quinolines / Vasodilation / Vascular Resistance / Penis / Lung / Vasoconstriction / Clinical Sciences / Lipopolysaccharides / Rats / Wistar Rats / Rabbits / Quinolines / Vasodilation / Vascular Resistance

New derivatives of 11-methyl-6-[2-(dimethylamino)ethyl]-6H-indolo[2,3-b]quinoline as cytotoxic DNA topoisomerase II inhibitors

Organic Chemistry / Cell Cycle / Humans / Mice / Animals / Male / Cell Proliferation / Quinolines / Human Fibroblasts / Structure activity Relationship / Antineoplastic Agents / Molecular Structure / Male / Cell Proliferation / Quinolines / Human Fibroblasts / Structure activity Relationship / Antineoplastic Agents / Molecular Structure

Montelukast exerts no acute direct effect on NO synthases

Gene expression / Humans / Female / Animals / Male / Penis / Lung / Vasoconstriction / Clinical Sciences / Lipopolysaccharides / Rats / Wistar Rats / Rabbits / Quinolines / Vasodilation / Vascular Resistance / Penis / Lung / Vasoconstriction / Clinical Sciences / Lipopolysaccharides / Rats / Wistar Rats / Rabbits / Quinolines / Vasodilation / Vascular Resistance

Neurotensin reduces glutamatergic transmission in the dorsolateral striatum via retrograde endocannabinoid signaling

Psychology / Neuropharmacology / Drug interactions / Synaptic Plasticity / Patch-clamp and imaging techniques / Signal Transduction / Dopamine / Glutamate / Habit Formation / Animals / Negative Feedback / dopamine receptor D4 / Synaptic Transmission / Neurons / Rats / Basal ganglia / Endocannabinoids / Pyrazoles / Quinolines / Neurosciences / Neurotensin / Intracellular Calcium / Piperidines / Phospholipase C / Signal Transduction / Dopamine / Glutamate / Habit Formation / Animals / Negative Feedback / dopamine receptor D4 / Synaptic Transmission / Neurons / Rats / Basal ganglia / Endocannabinoids / Pyrazoles / Quinolines / Neurosciences / Neurotensin / Intracellular Calcium / Piperidines / Phospholipase C

Using fragment cocktail crystallography to assist inhibitor design of Trypanosoma brucei nucleoside 2-deoxyribosyltransferase

Organic Chemistry / Medicinal Chemistry / Macromolecular X-Ray Crystallography / Animals / Trypanosoma brucei / Trypanosoma brucei brucei / Trypanocidal Agents / Amino Acid Sequence / Quinolines / Structure activity Relationship / Ligands / Molecular Structure / Trypanosoma brucei brucei / Trypanocidal Agents / Amino Acid Sequence / Quinolines / Structure activity Relationship / Ligands / Molecular Structure

Using fragment cocktail crystallography to assist inhibitor design of Trypanosoma brucei nucleoside 2-deoxyribosyltransferase

Organic Chemistry / Medicinal Chemistry / Macromolecular X-Ray Crystallography / Animals / Trypanosoma brucei / Trypanosoma brucei brucei / Trypanocidal Agents / Amino Acid Sequence / Quinolines / Structure activity Relationship / Ligands / Molecular Structure / Trypanosoma brucei brucei / Trypanocidal Agents / Amino Acid Sequence / Quinolines / Structure activity Relationship / Ligands / Molecular Structure

Development of CXCR3 antagonists. Part 4: Discovery of 2-amino-(4-tropinyl)quinolines

Organic Chemistry / Mice / Animals / Bioorganic and medicinal Chemistry / Quinolines / Biological Availability / Physicochemical Properties / Area Under Curve / Biological Availability / Physicochemical Properties / Area Under Curve
Copyright © 2017 DADOSPDF Inc.