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Thiazoles
Thiazoles
Quinolinium Salt as a Potent Inhibitor of Lymphocyte Apoptosis
Organic Chemistry / Apoptosis / Humans / Thiazoles / Lymphocytes / Salts / Toluene / Structure activity Relationship / Antineoplastic Agents / Glucocorticoids / Salts / Toluene / Structure activity Relationship / Antineoplastic Agents / Glucocorticoids
In vitro evaluation of bisnaphthalimidopropyl derivatives loaded into pegylated nanoparticles against Leishmania infantum protozoa
Medical Microbiology / Nanoparticles / Macrophages / Polymers / Cell line / Humans / Mice / Animals / Drug Delivery Systems / Quinolones / Antimicrobial agents / Leishmania infantum / Thiazoles / Drug Carriers / Lactic Acid / Cell Survival / Humans / Mice / Animals / Drug Delivery Systems / Quinolones / Antimicrobial agents / Leishmania infantum / Thiazoles / Drug Carriers / Lactic Acid / Cell Survival
Frontotemporal Dementia: Clinicopathological Correlations
Dementia / Immunohistochemistry / Neurodegenerative Diseases / Ubiquitin / Brain / Humans / Female / Male / Differential Diagnosis / Tauopathies / Clinical Sciences / Inclusion Bodies / Aged / Middle Aged / Adult / Frontotemporal Dementia / Annals / Thiazoles / Alzheimer Disease / Neurosciences / Age of Onset / Humans / Female / Male / Differential Diagnosis / Tauopathies / Clinical Sciences / Inclusion Bodies / Aged / Middle Aged / Adult / Frontotemporal Dementia / Annals / Thiazoles / Alzheimer Disease / Neurosciences / Age of Onset
Initial In Vitro Biological Response to Contemporary Endodontic Sealers
Dentistry / Water / Cell Culture / Mice / Animals / Ethanol / Sterilization / Epoxy Resins / Endodontics / Time Factors / Root Canal Filling Materials / Thiazoles / Polymethyl Methacrylates / Materials Testing / Acetone / Biocompatible Materials / Succinate Dehydrogenase / Solvents / Ethanol / Sterilization / Epoxy Resins / Endodontics / Time Factors / Root Canal Filling Materials / Thiazoles / Polymethyl Methacrylates / Materials Testing / Acetone / Biocompatible Materials / Succinate Dehydrogenase / Solvents
In vitro evaluation of bisnaphthalimidopropyl derivatives loaded into pegylated nanoparticles against Leishmania infantum protozoa
Medical Microbiology / Nanoparticles / Macrophages / Polymers / Cell line / Humans / Mice / Animals / Drug Delivery Systems / Quinolones / Antimicrobial agents / Leishmania infantum / Thiazoles / Drug Carriers / Lactic Acid / Cell Survival / Humans / Mice / Animals / Drug Delivery Systems / Quinolones / Antimicrobial agents / Leishmania infantum / Thiazoles / Drug Carriers / Lactic Acid / Cell Survival
ChemInform Abstract: Novel Design Principle Validated: Glucopyranosylidene-spiro-oxathiazole as New Nanomolar Inhibitor of Glycogen Phosphorylase, Potential Antidiabetic Agent
Organic Chemistry / Kinetics / Pharmaceutical Chemistry / Glucose / Animals / Drug Design / Oral Hypoglycemic Agents / Bioorganic and medicinal Chemistry / Rabbits / Thiazoles / Glycogen / Drug Design / Oral Hypoglycemic Agents / Bioorganic and medicinal Chemistry / Rabbits / Thiazoles / Glycogen
Frontotemporal dementia: Clinicopathological correlations
Dementia / Immunohistochemistry / Neurodegenerative Diseases / Ubiquitin / Brain / Humans / Female / Male / Differential Diagnosis / Tauopathies / Clinical Sciences / Inclusion Bodies / Aged / Middle Aged / Adult / Frontotemporal Dementia / Annals / Thiazoles / Alzheimer Disease / Neurosciences / Age of Onset / Humans / Female / Male / Differential Diagnosis / Tauopathies / Clinical Sciences / Inclusion Bodies / Aged / Middle Aged / Adult / Frontotemporal Dementia / Annals / Thiazoles / Alzheimer Disease / Neurosciences / Age of Onset
Indolic secondary metabolites protect Arabidopsis from the oomycete pathogen Phytophthora brassicae
Plant Biology / Plant diseases / Mutation / Disease resistance / Arabidopsis / Phytophthora / Sesquiterpenes / Thiazoles / Glucosinolates / Biochemistry and cell biology / Phytophthora / Sesquiterpenes / Thiazoles / Glucosinolates / Biochemistry and cell biology
Phenylacetic acid derivatives as hPPAR agonists
Organic Chemistry / Transcription Factors / Insulin Resistance / Blood Glucose / Mice / Animals / Male / Drug Design / Triglycerides / Rats / Oral Hypoglycemic Agents / Bioorganic and medicinal Chemistry / Thiazoles / Animals / Male / Drug Design / Triglycerides / Rats / Oral Hypoglycemic Agents / Bioorganic and medicinal Chemistry / Thiazoles
2,6-Diphenylthiazolo[3,2-b][1,2,4]triazoles as telomeric G-quadruplex stabilizers
Organic Chemistry / Macromolecular X-Ray Crystallography / Fluorescence Resonance Energy Transfer / Computer Simulation / Drug Design / Telomere / Triazoles / Thiazoles / Transition Temperature / Telomere / Triazoles / Thiazoles / Transition Temperature
In vitro activities of new and established triazoles against opportunistic filamentous and dimorphic fungi
Medical Microbiology / Fungi / Medical Mycology / Humans / Voriconazole / Antifungal Agents / Microbial Sensitivity Tests / Species Specificity / Triazoles / Thiazoles / Medical / Antifungal Agents / Microbial Sensitivity Tests / Species Specificity / Triazoles / Thiazoles / Medical
Novel selective thiazoleacetic acids as CRTH2 antagonists developed from in silico derived hits. Part 1
Organic Chemistry / Modeling / Prediction / Pharmacokinetics / Molecular modeling / Cercopithecus aethiops / Cell line / In Vitro / Humans / Animals / Resonant Energy Transfer / Bioluminescence / In Vivo / Rats / Molecular Model / Water Solubility / Acetic Acid / ADME / Bioorganic and medicinal Chemistry / Thiazoles / In Silico / Structure activity Relationship / Protein Binding / Chemical Synthesis / Selectivity / Binding affinity / Cercopithecus aethiops / Cell line / In Vitro / Humans / Animals / Resonant Energy Transfer / Bioluminescence / In Vivo / Rats / Molecular Model / Water Solubility / Acetic Acid / ADME / Bioorganic and medicinal Chemistry / Thiazoles / In Silico / Structure activity Relationship / Protein Binding / Chemical Synthesis / Selectivity / Binding affinity
Archazolid A-15- O -β- d -glucopyranoside and iso -Archazolid B: Potent V-ATPase Inhibitory Polyketides from the Myxobacteria Cystobacter violaceus and Archangium gephyra
Natural Products / Cytotoxicity / Structural Analysis / Biological Sciences / Cell line / In Vitro / Humans / Macrocycle / Mice / Female / Animals / Male / Bacteria / CHEMICAL SCIENCES / Isolation / Natural / Biological activity / Thiazoles / Antineoplastic Agents / Molecular Structure / Macrolides / In Vitro / Humans / Macrocycle / Mice / Female / Animals / Male / Bacteria / CHEMICAL SCIENCES / Isolation / Natural / Biological activity / Thiazoles / Antineoplastic Agents / Molecular Structure / Macrolides
Archazolid A-15-O-β-D-glucopyranoside and iso-Archazolid B: Potent V-ATPase Inhibitory Polyketides from the Myxobacteria Cystobacter violaceus and Archangium gephyra
Natural Products / Cytotoxicity / Structural Analysis / Biological Sciences / Cell line / In Vitro / Humans / Macrocycle / Mice / Female / Animals / Male / Bacteria / CHEMICAL SCIENCES / Isolation / Natural / Biological activity / Thiazoles / Antineoplastic Agents / Molecular Structure / Macrolides / In Vitro / Humans / Macrocycle / Mice / Female / Animals / Male / Bacteria / CHEMICAL SCIENCES / Isolation / Natural / Biological activity / Thiazoles / Antineoplastic Agents / Molecular Structure / Macrolides
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