Pharmacokinetics

Process Analytical Technology: A Review

Pharmacology / Pharmacy / Pharmacoepidemiology / Pharmacogenomics / Pharmaceutical Technology / Pharmacovigilance / Pharmacokinetics / Clinical Pharmacology / Pharmacy Practice / Pharmacognosy / Pharmacoeconomics / Pharmacognosy and Phytochemistry / Pharmaceutical Chemistry / Molecular Pharmacology / Herbal Pharmaceuticals / Pharmaceutical Analysis / Pharmaceutical Marketing / Pharmaceutics / Pharmaceutical Microbiology / Pharmaceutical industry / Pharmaceutical Biotechnology / Clinical Pharmacy / Pharmaceuticals / Pharmaceutical Sciences / Pharmaceutical / DOCTOR OF PHARMACY / Pharmacology and toxicology / Pharmaceutical formulation and development / Clinical Pharmacy Practice / Pharmacotherapy / Pharmaceutical Law / Pharmaceutical Formulation Technology / Pharmacovigilance / Pharmacokinetics / Clinical Pharmacology / Pharmacy Practice / Pharmacognosy / Pharmacoeconomics / Pharmacognosy and Phytochemistry / Pharmaceutical Chemistry / Molecular Pharmacology / Herbal Pharmaceuticals / Pharmaceutical Analysis / Pharmaceutical Marketing / Pharmaceutics / Pharmaceutical Microbiology / Pharmaceutical industry / Pharmaceutical Biotechnology / Clinical Pharmacy / Pharmaceuticals / Pharmaceutical Sciences / Pharmaceutical / DOCTOR OF PHARMACY / Pharmacology and toxicology / Pharmaceutical formulation and development / Clinical Pharmacy Practice / Pharmacotherapy / Pharmaceutical Law / Pharmaceutical Formulation Technology

Cyanopyridyl containing 1,4-dihydroindeno[1,2-c]pyrazoles as potent checkpoint kinase 1 inhibitors: Improving oral biovailability

Organic Chemistry / Hydrogen / Pharmacokinetics / DNA damage / Signal Transduction / In Vitro / Protein Kinases / Mice / Animals / Bioavailability / In Vivo / Rats / Pyridines / Bioorganic and medicinal Chemistry / Pyrazoles / Cyanides / Structure activity Relationship / Chemical Synthesis / Protein Kinase Inhibitors / Molecular Structure / In Vitro / Protein Kinases / Mice / Animals / Bioavailability / In Vivo / Rats / Pyridines / Bioorganic and medicinal Chemistry / Pyrazoles / Cyanides / Structure activity Relationship / Chemical Synthesis / Protein Kinase Inhibitors / Molecular Structure

Cyanopyridyl containing 1,4-dihydroindeno[1,2- c]pyrazoles as potent checkpoint kinase 1 inhibitors: Improving oral biovailability

Organic Chemistry / Hydrogen / Pharmacokinetics / DNA damage / Signal Transduction / In Vitro / Protein Kinases / Mice / Animals / Bioavailability / In Vivo / Rats / Pyridines / Bioorganic and medicinal Chemistry / Pyrazoles / Cyanides / Structure activity Relationship / Chemical Synthesis / Protein Kinase Inhibitors / Molecular Structure / In Vitro / Protein Kinases / Mice / Animals / Bioavailability / In Vivo / Rats / Pyridines / Bioorganic and medicinal Chemistry / Pyrazoles / Cyanides / Structure activity Relationship / Chemical Synthesis / Protein Kinase Inhibitors / Molecular Structure

Cyanopyridyl containing 1,4-dihydroindeno[1,2-c]pyrazoles as potent checkpoint kinase 1 inhibitors: Improving oral biovailability

Organic Chemistry / Hydrogen / Pharmacokinetics / DNA damage / Signal Transduction / In Vitro / Protein Kinases / Mice / Animals / Bioavailability / In Vivo / Rats / Pyridines / Bioorganic and medicinal Chemistry / Pyrazoles / Cyanides / Structure activity Relationship / Chemical Synthesis / Protein Kinase Inhibitors / Molecular Structure / In Vitro / Protein Kinases / Mice / Animals / Bioavailability / In Vivo / Rats / Pyridines / Bioorganic and medicinal Chemistry / Pyrazoles / Cyanides / Structure activity Relationship / Chemical Synthesis / Protein Kinase Inhibitors / Molecular Structure

Serial Magnetic Resonance Spectroscopy Reveals a Direct Metabolic Effect of Cediranib in Glioblastoma

Metabolism / Cancer / Pharmacokinetics / Magnetic Resonance Spectroscopy / Humans / Glioblastoma / Female / Male / Young Adult / Aged / Middle Aged / Adult / Brain Neoplasms / Quinazolines / Glioblastoma / Female / Male / Young Adult / Aged / Middle Aged / Adult / Brain Neoplasms / Quinazolines

Pharmacologic treatment can prevent pancreatic injury after ERCP: a meta-analysis

Pain / Clinical Trial / Statistical Analysis / Randomization / Pharmacokinetics / Treatment Outcome / Pancreatitis / Prevention / Somatostatin / Humans / Pancreas / Hormones / Statistical Significance / Acute Pancreatitis / Cost effectiveness / Metaanalysis / Randomized Trial / Meta Analysis / Publication Bias / Clinical Sciences / Gastrointestinal Endoscopy / Gastrointestinal / Endoscopic Retrograde Cholangiopancreatography / Acute Disease / Treatment Outcome / Pancreatitis / Prevention / Somatostatin / Humans / Pancreas / Hormones / Statistical Significance / Acute Pancreatitis / Cost effectiveness / Metaanalysis / Randomized Trial / Meta Analysis / Publication Bias / Clinical Sciences / Gastrointestinal Endoscopy / Gastrointestinal / Endoscopic Retrograde Cholangiopancreatography / Acute Disease

Novel selective thiazoleacetic acids as CRTH2 antagonists developed from in silico derived hits. Part 1

Organic Chemistry / Modeling / Prediction / Pharmacokinetics / Molecular modeling / Cercopithecus aethiops / Cell line / In Vitro / Humans / Animals / Resonant Energy Transfer / Bioluminescence / In Vivo / Rats / Molecular Model / Water Solubility / Acetic Acid / ADME / Bioorganic and medicinal Chemistry / Thiazoles / In Silico / Structure activity Relationship / Protein Binding / Chemical Synthesis / Selectivity / Binding affinity / Cercopithecus aethiops / Cell line / In Vitro / Humans / Animals / Resonant Energy Transfer / Bioluminescence / In Vivo / Rats / Molecular Model / Water Solubility / Acetic Acid / ADME / Bioorganic and medicinal Chemistry / Thiazoles / In Silico / Structure activity Relationship / Protein Binding / Chemical Synthesis / Selectivity / Binding affinity

A novel technique to monitor carboxypeptidase G2 expression in suicide gene therapy using 19 F magnetic resonance spectroscopy

Biomedical Engineering / Kinetics / Gene Therapy / Pharmacokinetics / Magnetic Resonance Spectroscopy / Molecular Imaging / Prodrugs / Humans / Nmr / Clinical Sciences / Fluorine / Buffers / Solutions / Molecular Imaging / Prodrugs / Humans / Nmr / Clinical Sciences / Fluorine / Buffers / Solutions

Pharmacologic treatment can prevent pancreatic injury after ERCP: a meta-analysis

Pain / Clinical Trial / Statistical Analysis / Randomization / Pharmacokinetics / Treatment Outcome / Pancreatitis / Prevention / Somatostatin / Humans / Pancreas / Hormones / Statistical Significance / Acute Pancreatitis / Cost effectiveness / Metaanalysis / Randomized Trial / Meta Analysis / Publication Bias / Clinical Sciences / Gastrointestinal Endoscopy / Gastrointestinal / Endoscopic Retrograde Cholangiopancreatography / Acute Disease / Treatment Outcome / Pancreatitis / Prevention / Somatostatin / Humans / Pancreas / Hormones / Statistical Significance / Acute Pancreatitis / Cost effectiveness / Metaanalysis / Randomized Trial / Meta Analysis / Publication Bias / Clinical Sciences / Gastrointestinal Endoscopy / Gastrointestinal / Endoscopic Retrograde Cholangiopancreatography / Acute Disease

Exposure-disease continuum for 2-chloro-2?-deoxyadenosine, a prototype ocular teratogen. 1. Dose-response analysis

Teratology / Pharmacokinetics / Immunohistochemistry / Mitochondria / Toxicity / Mutation / Mice / Animals / Eye / High Pressure Liquid Chromatography / Time Factors / Teratogens / Amino Acid Sequence / Base Sequence / Gestation / Molecular Sequence Data / Immunosuppressive Agents / Mutation / Mice / Animals / Eye / High Pressure Liquid Chromatography / Time Factors / Teratogens / Amino Acid Sequence / Base Sequence / Gestation / Molecular Sequence Data / Immunosuppressive Agents

Pharmacologic treatment can prevent pancreatic injury after ERCP: a meta-analysis

Pain / Clinical Trial / Statistical Analysis / Randomization / Pharmacokinetics / Treatment Outcome / Pancreatitis / Prevention / Somatostatin / Humans / Pancreas / Hormones / Statistical Significance / Acute Pancreatitis / Cost effectiveness / Metaanalysis / Randomized Trial / Meta Analysis / Publication Bias / Clinical Sciences / Gastrointestinal Endoscopy / Gastrointestinal / Endoscopic Retrograde Cholangiopancreatography / Acute Disease / Outcome measure / Adverse effect / Octreotide / Treatment Outcome / Pancreatitis / Prevention / Somatostatin / Humans / Pancreas / Hormones / Statistical Significance / Acute Pancreatitis / Cost effectiveness / Metaanalysis / Randomized Trial / Meta Analysis / Publication Bias / Clinical Sciences / Gastrointestinal Endoscopy / Gastrointestinal / Endoscopic Retrograde Cholangiopancreatography / Acute Disease / Outcome measure / Adverse effect / Octreotide

4-Amino-6-arylamino-pyrimidine-5-carbaldehyde hydrazones as potent ErbB-2/EGFR dual kinase inhibitors

Organic Chemistry / Modeling / Pharmacokinetics / Pharmaceutical Chemistry / Signal Transduction / Crystal structure / X Rays / In Vitro / Humans / Animals / Drug Design / Kinase inhibitor / Design Rationale / In Vivo / Hydrazones / Rats / Oximes / Molecular Model / Molecular Conformation / Bioorganic and medicinal Chemistry / Growth Factor / Structure activity Relationship / Chemical Synthesis / Protein Kinase Inhibitors / Receptor Tyrosine Kinase / Crystal structure / X Rays / In Vitro / Humans / Animals / Drug Design / Kinase inhibitor / Design Rationale / In Vivo / Hydrazones / Rats / Oximes / Molecular Model / Molecular Conformation / Bioorganic and medicinal Chemistry / Growth Factor / Structure activity Relationship / Chemical Synthesis / Protein Kinase Inhibitors / Receptor Tyrosine Kinase
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