Organic Chemistry

Bisbenzamidine isoxazoline derivatives as factor Xa inhibitors

Organic Chemistry / cerebral Venous sinus thrombosis / Blood Coagulation / Serine Protease

Bacterial diaminopimelate metabolism as a target for antibiotic design

Organic Chemistry / Bioorganic and medicinal Chemistry

3-Amino-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazoles: A new class of CDK2 inhibitors

Organic Chemistry / Enzyme Inhibitors / Macromolecular X-Ray Crystallography / Humans / Bioorganic and medicinal Chemistry / Cell Proliferation / Pyrazoles / Aurora kinases / Structure activity Relationship / Antineoplastic Agents / Molecular Structure / Cell Proliferation / Pyrazoles / Aurora kinases / Structure activity Relationship / Antineoplastic Agents / Molecular Structure

Indole-2-carboxamides as novel NR2B selective NMDA receptor antagonists

Organic Chemistry / Magnetic Resonance Spectroscopy / Phenols / Radioligand Assay / Bioorganic and medicinal Chemistry / Biological activity / Structure activity Relationship / Piperidines / Biological activity / Structure activity Relationship / Piperidines

Benzimidazole-2-carboxamides as novel NR2B selective NMDA receptor antagonists

Organic Chemistry / Amides / Bioorganic and medicinal Chemistry / Biological activity / Benzimidazoles / Structure activity Relationship / Molecular Structure / Formalin Test / Structure activity Relationship / Molecular Structure / Formalin Test

Oxamides as novel NR2B selective NMDA receptor antagonists

Organic Chemistry / Mice / Animals / Bioorganic and medicinal Chemistry / Structure activity Relationship / Molecular Structure / Formalin Test / Molecular Structure / Formalin Test

THE ATACAMA COSMOLOGY TELESCOPE: COSMOLOGICAL PARAMETERS FROM THE 2008 POWER SPECTRUM

Organic Chemistry / Astrophysical Plasma / Kinetics / Parameter estimation / Cosmic Microwave Background / Seasonality / Spectrum / Infrared / Power Spectrum / Analytical Model / Indexation / Cosmic Microwave Background Radiation / Cosmic String / Scale Invariance / Seasonality / Spectrum / Infrared / Power Spectrum / Analytical Model / Indexation / Cosmic Microwave Background Radiation / Cosmic String / Scale Invariance

Potent 4-amino-5-azaindole factor VIIa inhibitors

Organic Chemistry / Pyridines / Bioorganic and medicinal Chemistry / Structure activity Relationship / Serine Protease / Tissue Factor / Molecular Structure / Tissue Factor / Molecular Structure

Silvestrol and Episilvestrol, Potential Anticancer Rocaglate Derivatives from Aglaia silvestris

Inorganic Chemistry / Organic Chemistry / Humans / Mice / Animals / Vascular endothelium / The / KB cells / Molecular Structure / Triterpenes / Aglaia / Vascular endothelium / The / KB cells / Molecular Structure / Triterpenes / Aglaia

N-Caffeoylphenalkylamide derivatives as bacterial efflux pump inhibitors

Organic Chemistry / Multidrug Resistance / Natural Product / Bacteria / Staphylococcus aureus / Membrane transport proteins / Anti-Bacterial Agents / Plant extracts / Amides / Microbial Sensitivity Tests / Reserpine / Structure activity Relationship / Norfloxacin / Membrane transport proteins / Anti-Bacterial Agents / Plant extracts / Amides / Microbial Sensitivity Tests / Reserpine / Structure activity Relationship / Norfloxacin

Fluorogenic ester substrates to assess proteolytic activity

Organic Chemistry / Kinetics / Substrate Specificity / Enzymatic Activity / Esters / Molecular Structure / Fluorescein / Molecular Structure / Fluorescein

Tailor-made Oligosilyl Potassium Compounds

Inorganic Chemistry / Organic Chemistry / Organometallics / Potassium

N-1H-Benzimidazol-5-ylbenzenesulfonamide derivatives as potent hPXR agonists

Organic Chemistry / Drug metabolism / Nuclear Receptor / Cell line / Humans / Drug Design / Enzyme / Bioorganic and medicinal Chemistry / Primary Culture / Benzimidazoles / Human Disease / Structure activity Relationship / Chemical Modification / Molecular Structure / Gene Expression Regulation / Pregnane X Receptor / Drug Design / Enzyme / Bioorganic and medicinal Chemistry / Primary Culture / Benzimidazoles / Human Disease / Structure activity Relationship / Chemical Modification / Molecular Structure / Gene Expression Regulation / Pregnane X Receptor
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