Organic Chemistry

Biosynthesis of Zeaxanthin via Mevalonate in Paracoccus Species Strain PTA-3335. A Product-Based Retrobiosynthetic Study †

Inorganic Chemistry / Organic Chemistry / Magnetic Resonance Spectroscopy / The / Beta Carotene / Molecular Structure

Biosynthesis of Zeaxanthin via Mevalonate in Paracoccus Species Strain PTA-3335. A Product-Based Retrobiosynthetic Study †

Inorganic Chemistry / Organic Chemistry / Magnetic Resonance Spectroscopy / The / Beta Carotene / Molecular Structure

Essential Oils of Micromeria dalmatica Benth ., a Balkan Endemic Species of Section Pseudomelissa

Organic Chemistry / Principal Component Analysis / Lamiaceae / Gas Chromatography/mass Spectrometry / Balkan Peninsula

2,6-Diphenylthiazolo[3,2-b][1,2,4]triazoles as telomeric G-quadruplex stabilizers

Organic Chemistry / Macromolecular X-Ray Crystallography / Fluorescence Resonance Energy Transfer / Computer Simulation / Drug Design / Telomere / Triazoles / Thiazoles / Transition Temperature / Telomere / Triazoles / Thiazoles / Transition Temperature

Antitrypanosomal Cycloartane Glycosides fromAstragalus baibutensis

Organic Chemistry / Magnetic Resonance Spectroscopy / Animals / Terpenes / Trypanosoma / Glycosides / Molecular Structure / Triterpenes / Glycosides / Molecular Structure / Triterpenes

Palmerolide macrolides from the Antarctic tunicate Synoicum adareanum

Organic Chemistry / Humans / Melanoma / Animals / Natural Product / Cattle / Cytotoxic Activity / Molecular Conformation / Bioorganic and medicinal Chemistry / Antineoplastic Agents / Macrolides / Cattle / Cytotoxic Activity / Molecular Conformation / Bioorganic and medicinal Chemistry / Antineoplastic Agents / Macrolides

Imidazo-pyrazine derivatives as potent CXCR3 antagonists

Organic Chemistry / Lung Inflammation / Humans / Mice / Animals / Anti-inflammatory agents / Rats / Molecular Conformation / Bioorganic and medicinal Chemistry / Imidazoles / Anti-inflammatory agents / Rats / Molecular Conformation / Bioorganic and medicinal Chemistry / Imidazoles

Iodo bis bistrimethylsilylamido lanthanides

Inorganic Chemistry / Organic Chemistry / Organometallic Chemistry / Potassium

Cyanopyridyl containing 1,4-dihydroindeno[1,2-c]pyrazoles as potent checkpoint kinase 1 inhibitors: Improving oral biovailability

Organic Chemistry / Hydrogen / Pharmacokinetics / DNA damage / Signal Transduction / In Vitro / Protein Kinases / Mice / Animals / Bioavailability / In Vivo / Rats / Pyridines / Bioorganic and medicinal Chemistry / Pyrazoles / Cyanides / Structure activity Relationship / Chemical Synthesis / Protein Kinase Inhibitors / Molecular Structure / In Vitro / Protein Kinases / Mice / Animals / Bioavailability / In Vivo / Rats / Pyridines / Bioorganic and medicinal Chemistry / Pyrazoles / Cyanides / Structure activity Relationship / Chemical Synthesis / Protein Kinase Inhibitors / Molecular Structure

Cyanopyridyl containing 1,4-dihydroindeno[1,2- c]pyrazoles as potent checkpoint kinase 1 inhibitors: Improving oral biovailability

Organic Chemistry / Hydrogen / Pharmacokinetics / DNA damage / Signal Transduction / In Vitro / Protein Kinases / Mice / Animals / Bioavailability / In Vivo / Rats / Pyridines / Bioorganic and medicinal Chemistry / Pyrazoles / Cyanides / Structure activity Relationship / Chemical Synthesis / Protein Kinase Inhibitors / Molecular Structure / In Vitro / Protein Kinases / Mice / Animals / Bioavailability / In Vivo / Rats / Pyridines / Bioorganic and medicinal Chemistry / Pyrazoles / Cyanides / Structure activity Relationship / Chemical Synthesis / Protein Kinase Inhibitors / Molecular Structure

Novel Antibacterial Class:  A Series of Tetracyclic Derivatives

Organic Chemistry / Medicinal Chemistry / Streptococcus pneumoniae / Humans / Anti-Bacterial Agents / Medicinal / Microbial Sensitivity Tests / B Lymphocytes / Structure activity Relationship / Protein Biosynthesis / Medicinal / Microbial Sensitivity Tests / B Lymphocytes / Structure activity Relationship / Protein Biosynthesis

Using fragment cocktail crystallography to assist inhibitor design of Trypanosoma brucei nucleoside 2-deoxyribosyltransferase

Organic Chemistry / Medicinal Chemistry / Macromolecular X-Ray Crystallography / Animals / Trypanosoma brucei / Trypanosoma brucei brucei / Trypanocidal Agents / Amino Acid Sequence / Quinolines / Structure activity Relationship / Ligands / Molecular Structure / Trypanosoma brucei brucei / Trypanocidal Agents / Amino Acid Sequence / Quinolines / Structure activity Relationship / Ligands / Molecular Structure

Cyanopyridyl containing 1,4-dihydroindeno[1,2-c]pyrazoles as potent checkpoint kinase 1 inhibitors: Improving oral biovailability

Organic Chemistry / Hydrogen / Pharmacokinetics / DNA damage / Signal Transduction / In Vitro / Protein Kinases / Mice / Animals / Bioavailability / In Vivo / Rats / Pyridines / Bioorganic and medicinal Chemistry / Pyrazoles / Cyanides / Structure activity Relationship / Chemical Synthesis / Protein Kinase Inhibitors / Molecular Structure / In Vitro / Protein Kinases / Mice / Animals / Bioavailability / In Vivo / Rats / Pyridines / Bioorganic and medicinal Chemistry / Pyrazoles / Cyanides / Structure activity Relationship / Chemical Synthesis / Protein Kinase Inhibitors / Molecular Structure

Synthesis of potassium (2R)-2-O-α-d-glucopyranosyl-(1→6)-α-d-glucopyranosyl-2,3-dihydroxypropanoate a natural compatible solute

Organic Chemistry / Glycosylation / Carbohydrate / Biochemistry and cell biology / Molecular Structure
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